PDB Information

PDB5Z0S
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Based Discovery of a Series of 5H-Pyrrolo[2,3-b]pyrazine FGFR Kinase Inhibitors
Jiang, A., Liu, Q., Wang, R., Wei, P., Dai, Y., Wang, X., Xu, Y., Ma, Y., Ai, J., Shen, J., Ding, J., Xiong, B.
Molecules
HeaderTransferase/Transferase Inhibitor
Released2017-12-20
Resolution2.450
CATH Insert Date30 Dec, 2018

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 30 Dec, 2018 Chopped
B 30 Dec, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5z0sA01 31 Dec, 2018 3.30.200.20 Assigned
5z0sA02 31 Dec, 2018 1.10.510.10 Assigned
5z0sB01 31 Dec, 2018 3.30.200.20 Assigned
5z0sB02 31 Dec, 2018 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P11362 FGFR1_HUMAN Homo sapiens Fibroblast growth factor receptor 1
P11362 FGFR1_HUMAN Homo sapiens Fibroblast growth factor receptor 1