PDB Information

PDB5YOV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups.
Hu, J., Wang, Y., Li, Y., Cao, D., Xu, L., Song, S., Damaneh, M.S., Li, J., Chen, Y., Wang, X., Chen, L., Shen, J., Miao, Z., Xiong, B.
Eur.J.Med.Chem.
HeaderTranscription/Inhibitor
Released2017-10-31
Resolution1.450
CATH Insert Date16 Dec, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5yovA01 28 Feb, 2019 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4