PDB 5yov
PDB Information
| PDB | 5YOV |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups.
Eur.J.Med.Chem.
|
| Header | Transcription/Inhibitor |
| Released | 2017-10-31 |
| Resolution | 1.450 |
| CATH Insert Date | 16 Dec, 2018 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Dec, 2018 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5yovA01 | 28 Feb, 2019 | 1.20.920.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
