PDB Information

PDB5YJO
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Irreversible Inhibitors Targeting Histone Methyltransferase, SMYD3.
Huang, C., Liew, S.S., Lin, G.R., Poulsen, A., Ang, M.J.Y., Chia, B.C.S., Chew, S.Y., Kwek, Z.P., Wee, J.L.K., Ong, E.H., Retna, P., Baburajendran, N., Li, R., Yu, W., Koh-Stenta, X., Ngo, A., Manesh, S., Fulwood, J., Ke, Z., Chung, H.H., Sepramaniam, S., Chew, X.H., Dinie, N., Lee, M.A., Chew, Y.S., Low, C.B., Pendharkar, V., Manoharan, V., Vuddagiri, S., Sangthongpitag, K., Joy, J., Matter, A., Hill, J., Keller, T.H., Foo, K.
Acs Med.Chem.Lett.
HeaderTransferase/Inhibitor
Released2017-10-11
Resolution2.140
CATH Insert Date16 Dec, 2018

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Dec, 2018 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5yjoA01 27 Feb, 2019 2.170.270.10 Assigned
5yjoA02 27 Feb, 2019 6.10.140.2220 Assigned
5yjoA03 27 Feb, 2019 1.10.220.160 Assigned
5yjoA04 27 Feb, 2019 1.25.40.970 Assigned
5yjoA05 27 Feb, 2019 1.25.40.10 Assigned

UniProtKB Entries (0)

Accession Gene ID Taxon Description