PDB 5y8y

PDB Links
Overview

PDB Information

PDB	5Y8Y
Method	X-RAY DIFFRACTION
Host Organism	Escherichia coli BL21
Gene Source	Homo sapiens
Primary Citation	Structure-Based Discovery and Optimization of Benzo[ d]isoxazole Derivatives as Potent and Selective BET Inhibitors for Potential Treatment of Castration-Resistant Prostate Cancer (CRPC) Zhang, M., Zhang, Y., Song, M., Xue, X., Wang, J., Wang, C., Zhang, C., Li, C., Xiang, Q., Zou, L., Wu, X., Wu, C., Dong, B., Xue, W., Zhou, Y., Chen, H., Wu, D., Ding, K., Xu, Y. J. Med. Chem.
Header	Transcription
Released	2017-08-21
Resolution	1.870
CATH Insert Date	06 Jul, 2018

PDB Images (3)

Image of CATH 5y8y

5y8y

PDB 5y8y

Image of CATH 5y8yA

5y8yA

PDB Chain 5y8yA

Image of CATH 5y8yA01

5y8yA01

CATH Domain 5y8yA01

PDB Prints

PDB Chains (1)

Chain ID	Date inserted into CATH	CATH Status
A	06 Jul, 2018	Chopped

CATH Domains (1)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
5y8yA01	19 Jul, 2018	1.20.920.10	Assigned

UniProtKB Entries (1)

Accession	Gene ID	Taxon	Description
O60885	BRD4_HUMAN	Homo sapiens	Bromodomain-containing protein 4