PDB Information

PDB5XUI
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors.
Chino, A., Seo, R., Amano, Y., Namatame, I., Hamaguchi, W., Honbou, K., Mihara, T., Yamazaki, M., Tomishima, M., Masuda, N.
Chem. Pharm. Bull.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-06-23
Resolution2.770
CATH Insert Date03 Jun, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5xuiA00 28 Jun, 2018 1.10.1300.10 Assigned
5xuiB00 28 Jun, 2018 1.10.1300.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9Y233 PDE10_HUMAN Homo sapiens cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
Q9Y233 PDE10_HUMAN Homo sapiens cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A