PDB 5xsr
PDB Information
| PDB | 5XSR |
| Method | X-RAY DIFFRACTION |
| Host Organism | Enterobacteria phage L1 |
| Gene Source | Homo sapiens |
| Primary Citation | Design and synthesis of 2-(4,5,6,7-tetrahydrothienopyridin-2-yl)-benzoimidazole carboxamides as novel orally efficacious Poly(ADP-ribose)polymerase (PARP) inhibitors
Eur J Med Chem
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2017-06-15 |
| Resolution | 2.300 |
| CATH Insert Date | 03 Jun, 2018 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 03 Jun, 2018 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5xsrA01 | 28 Jun, 2018 | Holding pen | |
| 5xsrA02 | 28 Jun, 2018 | 3.90.228.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P09874 | PARP1_HUMAN | Homo sapiens | Poly [ADP-ribose] polymerase 1 |
