PDB Information

PDB5XMX
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Novel highly selective peroxisome proliferator-activated receptor delta (PPAR delta) modulators with pharmacokinetic properties suitable for once-daily oral dosing.
Lagu, B., Kluge, A.F., Fredenburg, R.A., Tozzo, E., Senaiar, R.S., Jaleel, M., Panigrahi, S.K., Tiwari, N.K., Krishnamurthy, N.R., Takahashi, T., Patane, M.A.
Bioorg. Med. Chem. Lett.
HeaderTranscription/Inhibitor
Released2017-05-16
Resolution2.000
CATH Insert Date03 Jun, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5xmxA00 28 Jun, 2018 1.10.565.10 Assigned
5xmxB00 28 Jun, 2018 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q03181 PPARD_HUMAN Homo sapiens Peroxisome proliferator-activated receptor delta
Q03181 PPARD_HUMAN Homo sapiens Peroxisome proliferator-activated receptor delta