PDB Information

PDB5WI1
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHomo sapiens
Primary Citation
Fragment-based discovery of a potent NAMPT inhibitor.
Korepanova, A., Longenecker, K.L., Pratt, S.D., Panchal, S.C., Clark, R.F., Lake, M., Gopalakrishnan, S.M., Raich, D., Sun, C., Petros, A.M.
Bioorg. Med. Chem. Lett.
HeaderTransferase/Transferase Inhibitor
Released2017-07-18
Resolution1.990
CATH Insert Date03 Jun, 2018

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5wi1A01 28 Jun, 2018 Holding pen
5wi1A02 28 Jun, 2018 3.20.20.70 Assigned
5wi1B01 28 Jun, 2018 Holding pen
5wi1B02 28 Jun, 2018 3.20.20.70 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P43490 NAMPT_HUMAN Homo sapiens Nicotinamide phosphoribosyltransferase
P43490 NAMPT_HUMAN Homo sapiens Nicotinamide phosphoribosyltransferase