PDB Information

PDB5WBE
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceOvis aries
Primary Citation
Structural basis for selective inhibition of Cyclooxygenase-1 (COX-1) by diarylisoxazoles mofezolac and 3-(5-chlorofuran-2-yl)-5-methyl-4-phenylisoxazole (P6).
Cingolani, G., Panella, A., Perrone, M.G., Vitale, P., Di Mauro, G., Fortuna, C.G., Armen, R.S., Ferorelli, S., Smith, W.L., Scilimati, A.
Eur J Med Chem
HeaderOxidoreductase/Oxidoreductase Inhibitor
Released2017-06-28
Resolution2.750
CATH Insert Date14 Nov, 2017

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5wbeA01 10 Dec, 2017 2.10.25.10 Assigned
5wbeA02 10 Dec, 2017 1.10.640.10 Assigned
5wbeB01 10 Dec, 2017 2.10.25.10 Assigned
5wbeB02 10 Dec, 2017 1.10.640.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P05979 PGH1_SHEEP Ovis aries Prostaglandin G/H synthase 1
P05979 PGH1_SHEEP Ovis aries Prostaglandin G/H synthase 1