PDB 5w4w
PDB Information
| PDB | 5W4W |
| Method | X-RAY DIFFRACTION |
| Host Organism | Insect cell expression vector pTIE1 |
| Gene Source | Homo sapiens |
| Primary Citation | Identification and Profiling of a Selective and Brain Penetrant Radioligand for in Vivo Target Occupancy Measurement of Casein Kinase 1 (CK1) Inhibitors.
ACS Chem Neurosci
|
| Header | Transferase/Inhibitor |
| Released | 2017-06-13 |
| Resolution | 1.990 |
| CATH Insert Date | 14 Nov, 2017 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 14 Nov, 2017 | Chopped |
| B | 14 Nov, 2017 | Chopped |
| C | 14 Nov, 2017 | Chopped |
| D | 14 Nov, 2017 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5w4wA01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
| 5w4wA02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
| 5w4wB01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
| 5w4wB02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
| 5w4wC01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
| 5w4wC02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
| 5w4wD01 | 10 Dec, 2017 | 3.30.200.20 | Assigned |
| 5w4wD02 | 10 Dec, 2017 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
| P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
| P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
| P48730 | KC1D_HUMAN | Homo sapiens | Casein kinase I isoform delta |
