PDB Information

PDB5VSK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Guided Development of a Potent and Selective Non-covalent Active-Site Inhibitor of USP7.
Lamberto, I., Liu, X., Seo, H.S., Schauer, N.J., Iacob, R.E., Hu, W., Das, D., Mikhailova, T., Weisberg, E.L., Engen, J.R., Anderson, K.C., Chauhan, D., Dhe-Paganon, S., Buhrlage, S.J.
Cell Chem Biol
HeaderHydrolase/Hydrolase Inhibitor
Released2017-05-11
Resolution3.330
CATH Insert Date07 Jan, 2018

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Jan, 2018 Chopped
B 07 Jan, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5vskA01 05 May, 2018 Holding pen
5vskA02 05 May, 2018 2.20.210.10 Assigned
5vskA03 05 May, 2018 Holding pen
5vskB00 05 May, 2018 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q93009 UBP7_HUMAN Homo sapiens Ubiquitin carboxyl-terminal hydrolase 7
Q93009 UBP7_HUMAN Homo sapiens Ubiquitin carboxyl-terminal hydrolase 7