PDB Information

PDB5VSF
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-activity relationship studies of G9a-like protein (GLP) inhibitors.
Xiong, Y., Li, F., Babault, N., Wu, H., Dong, A., Zeng, H., Chen, X., Arrowsmith, C.H., Brown, P.J., Liu, J., Vedadi, M., Jin, J.
Bioorg. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2017-05-11
Resolution1.700
CATH Insert Date14 Nov, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5vsfA00 10 Dec, 2017 2.170.270.10 Assigned
5vsfB00 10 Dec, 2017 2.170.270.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H9B1 EHMT1_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT1
Q9H9B1 EHMT1_HUMAN Homo sapiens Histone-lysine N-methyltransferase EHMT1