PDB 5vrp
PDB Information
PDB | 5VRP |
Method | X-RAY DIFFRACTION |
Host Organism | Homo sapiens |
Gene Source | Homo sapiens |
Primary Citation | Discovery of renin inhibitors containing a simple aspartate binding moiety that imparts reduced P450 inhibition.
Bioorg. Med. Chem. Lett.
|
Header | Hydrolase/Hydrolase Inhibitor |
Released | 2017-05-11 |
Resolution | 3.220 |
CATH Insert Date | 14 Nov, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 14 Nov, 2017 | Chopped |
B | 14 Nov, 2017 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5vrpA01 | 10 Dec, 2017 | 2.40.70.10 | Assigned |
5vrpA02 | 10 Dec, 2017 | 2.40.70.10 | Assigned |
5vrpB01 | 10 Dec, 2017 | 2.40.70.10 | Assigned |
5vrpB02 | 10 Dec, 2017 | 2.40.70.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P00797 | RENI_HUMAN | Homo sapiens | Renin |
P00797 | RENI_HUMAN | Homo sapiens | Renin |