PDB Information

PDB5VO1
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
Selective Inhibitors of Dual Leucine Zipper Kinase (DLK, MAP3K12) with Activity in a Model of Alzheimer's Disease.
Patel, S., Meilandt, W.J., Erickson, R.I., Chen, J., Deshmukh, G., Estrada, A.A., Fuji, R.N., Gibbons, P., Gustafson, A., Harris, S.F., Imperio, J., Liu, W., Liu, X., Liu, Y., Lyssikatos, J.P., Ma, C., Yin, J., Lewcock, J.W., Siu, M.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2017-05-01
Resolution2.450
CATH Insert Date14 Nov, 2017

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5vo1A01 10 Dec, 2017 3.30.200.20 Assigned
5vo1A02 10 Dec, 2017 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q12852 M3K12_HUMAN Homo sapiens Mitogen-activated protein kinase kinase kinase 12