Discovery of Potent and Selective Tricyclic Inhibitors of Bruton's Tyrosine Kinase with Improved Druglike Properties.
Wang, X., Barbosa, J., Blomgren, P., Bremer, M.C., Chen, J., Crawford, J.J., Deng, W., Dong, L., Eigenbrot, C., Gallion, S., Hau, J., Hu, H., Johnson, A.R., Katewa, A., Kropf, J.E., Lee, S.H., Liu, L., Lubach, J.W., Macaluso, J., Maciejewski, P., Mitchell, S.A., Ortwine, D.F., DiPaolo, J., Reif, K., Scheerens, H., Schmitt, A., Wong, H., Xiong, J.M., Xu, J., Zhao, Z., Zhou, F., Currie, K.S., Young, W.B.
ACS Med Chem Lett