PDB 5v82

PDB Information

PDB5V82
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of 5-Azaindazole (GNE-955) as a Potent Pan-Pim Inhibitor with Optimized Bioavailability.
Wang, X., Kolesnikov, A., Tay, S., Chan, G., Chao, Q., Do, S., Drummond, J., Ebens, A.J., Liu, N., Ly, J., Harstad, E., Hu, H., Moffat, J., Munugalavadla, V., Murray, J., Slaga, D., Tsui, V., Volgraf, M., Wallweber, H., Chang, J.H.
J. Med. Chem.
HeaderTransferase/Inhibitor
Released2017-03-21
Resolution1.890
CATH Insert Date14 May, 2017

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 15 May, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5v82A01 06 Nov, 2017 3.30.200.20 Assigned
5v82A02 06 Nov, 2017 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1