PDB Information

PDB5V71
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli K-12
Gene SourceHomo sapiens
Primary Citation
KRAS G12C Drug Development: Discrimination between Switch II Pocket Configurations Using Hydrogen/Deuterium-Exchange Mass Spectrometry.
Lu, J., Harrison, R.A., Li, L., Zeng, M., Gondi, S., Scott, D., Gray, N.S., Engen, J.R., Westover, K.D.
Structure
HeaderHydrolase/Hydrolase Inhibitor
Released2017-03-17
Resolution2.230
CATH Insert Date14 Nov, 2017

PDB Images (13)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped
C 14 Nov, 2017 Chopped
D 14 Nov, 2017 Chopped
E 14 Nov, 2017 Chopped
F 14 Nov, 2017 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
5v71A00 10 Dec, 2017 3.40.50.300 Assigned
5v71B00 10 Dec, 2017 3.40.50.300 Assigned
5v71C00 10 Dec, 2017 3.40.50.300 Assigned
5v71D00 10 Dec, 2017 3.40.50.300 Assigned
5v71E00 10 Dec, 2017 3.40.50.300 Assigned
5v71F00 10 Dec, 2017 3.40.50.300 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas
P01116 RASK_HUMAN Homo sapiens GTPase KRas