PDB Information

PDB5V61
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Guided Strategy for the Development of Potent Bivalent ERK Inhibitors.
Lechtenberg, B.C., Mace, P.D., Sessions, E.H., Williamson, R., Stalder, R., Wallez, Y., Roth, G.P., Riedl, S.J., Pasquale, E.B.
ACS Med Chem Lett
HeaderTransferase/Inhibitor
Released2017-03-15
Resolution2.200
CATH Insert Date14 Nov, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
I 14 Nov, 2017 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5v61A01 10 Dec, 2017 3.30.200.20 Assigned
5v61A02 10 Dec, 2017 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P28482 MK01_HUMAN Homo sapiens Mitogen-activated protein kinase 1
Q15418 KS6A1_HUMAN Homo sapiens Ribosomal protein S6 kinase alpha-1