PDB Information

PDB5UVC
MethodX-RAY DIFFRACTION
Host OrganismBaculovirus expression vector pFastBac1-HM
Gene SourceHomo sapiens
Primary Citation
Design, Synthesis, and Evaluation of the Highly Selective and Potent G-Protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor for the Potential Treatment of Heart Failure.
Okawa, T., Aramaki, Y., Yamamoto, M., Kobayashi, T., Fukumoto, S., Toyoda, Y., Henta, T., Hata, A., Ikeda, S., Kaneko, M., Hoffman, I.D., Sang, B.C., Zou, H., Kawamoto, T.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2017-02-20
Resolution2.650
CATH Insert Date14 Nov, 2017

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P25098 ARBK1_HUMAN Homo sapiens Beta-adrenergic receptor kinase 1