PDB Information

PDB5UPJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 2
Primary Citation
Use of medium-sized cycloalkyl rings to enhance secondary binding: discovery of a new class of human immunodeficiency virus (HIV) protease inhibitors.
Romines, K.R., Watenpaugh, K.D., Tomich, P.K., Howe, W.J., Morris, J.K., Lovasz, K.D., Mulichak, A.M., Finzel, B.C., Lynn, J.C., Horng, M.-M., Schwende, F.J., Ruwart, M.J., Zipp, G.L., Chong, K.-T., Dolak, L.A., Toth, L.N., Howard, G.M., Rush, B.D., Wilkinson, K.F., Possert, P.L., Dalga, R.J., Hinshaw, R.R.
J.Med.Chem.
HeaderHydrolase
Released1996-12-10
Resolution2.300
CATH Insert Date05 Mar, 2006

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Mar, 2006 Chopped
B 05 Mar, 2006 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5upjA00 05 Mar, 2006 2.40.70.10 Assigned
5upjB00 05 Mar, 2006 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P04584 POL_HV2RO Human immunodeficiency virus type 2 (ISOLATE ROD) Gag-Pol polyprotein
P04584 POL_HV2RO Human immunodeficiency virus type 2 (ISOLATE ROD) Gag-Pol polyprotein