PDB Information

PDB5ULT
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Design and Development of Highly Potent HIV-1 Protease Inhibitors with a Crown-Like Oxotricyclic Core as the P2-Ligand To Combat Multidrug-Resistant HIV Variants.
Ghosh, A.K., Rao, K.V., Nyalapatla, P.R., Osswald, H.L., Martyr, C.D., Aoki, M., Hayashi, H., Agniswamy, J., Wang, Y.F., Bulut, H., Das, D., Weber, I.T., Mitsuya, H.
J. Med. Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2017-01-25
Resolution1.530
CATH Insert Date14 May, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 15 May, 2017 Chopped
B 15 May, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5ultA00 06 Nov, 2017 2.40.70.10 Assigned
5ultB00 06 Nov, 2017 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P03366 POL_HV1B1 Human immunodeficiency virus type 1 BH10 Gag-Pol polyprotein
P03366 POL_HV1B1 Human immunodeficiency virus type 1 BH10 Gag-Pol polyprotein