PDB Information

PDB5UKJ
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
Rationally Designed PI3K alpha Mutants to Mimic ATR and Their Use to Understand Binding Specificity of ATR Inhibitors.
Lu, Y., Knapp, M., Crawford, K., Warne, R., Elling, R., Yan, K., Doyle, M., Pardee, G., Zhang, L., Ma, S., Mamo, M., Ornelas, E., Pan, Y., Bussiere, D., Jansen, J., Zaror, I., Lai, A., Barsanti, P., Sim, J.
J. Mol. Biol.
HeaderTransferase/Signaling Protein/Inhibitor
Released2017-01-23
Resolution2.800
CATH Insert Date14 May, 2017

PDB Images (3)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 15 May, 2017 Holding pen
B 15 May, 2017 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P42336 PK3CA_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
P27986 P85A_HUMAN Homo sapiens Phosphatidylinositol 3-kinase regulatory subunit alpha