PDB 5ubt
PDB Information
| PDB | 5UBT |
| Method | X-RAY DIFFRACTION |
| Host Organism | unidentified baculovirus |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine derivatives as highly potent and selective PI3K delta inhibitors.
Bioorg. Med. Chem. Lett.
|
| Header | Transferase/Transferase Regulator |
| Released | 2016-12-21 |
| Resolution | 2.830 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (3)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Holding pen |
| B | 08 May, 2017 | Holding pen |
CATH Domains (0)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O00329 | PK3CD_HUMAN | Homo sapiens | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform |
| P27986 | P85A_HUMAN | Homo sapiens | Phosphatidylinositol 3-kinase regulatory subunit alpha |
