PDB 5u6v

PDB Information

PDB5U6V
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design, Synthesis, and Biological Activity of 1,2,3-Triazolobenzodiazepine BET Bromodomain Inhibitors.
Sharp, P.P., Garnier, J.M., Hatfaludi, T., Xu, Z., Segal, D., Jarman, K.E., Jousset, H., Garnham, A., Feutrill, J.T., Cuzzupe, A., Hall, P., Taylor, S., Walkley, C.R., Tyler, D., Dawson, M.A., Czabotar, P., Wilks, A.F., Glaser, S., Huang, D.C.S., Burns, C.J.
ACS Med Chem Lett
HeaderTranscription/Transcription Inhibitor
Released2016-12-09
Resolution1.780
CATH Insert Date07 Jan, 2018

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Jan, 2018 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5u6vA00 11 Jan, 2018 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P25440 BRD2_HUMAN Homo sapiens Bromodomain-containing protein 2