PDB Information

PDB5U6E
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Synthesis, Antiviral Potency, in Vitro ADMET, and X-ray Structure of Potent CD4 Mimics as Entry Inhibitors That Target the Phe43 Cavity of HIV-1 gp120.
Curreli, F., Kwon, Y.D., Belov, D.S., Ramesh, R.R., Kurkin, A.V., Altieri, A., Kwong, P.D., Debnath, A.K.
J. Med. Chem.
HeaderViral Protein
Released2016-12-07
Resolution2.100
CATH Insert Date07 May, 2017

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5u6eA01 23 May, 2017 2.170.40.20 Assigned
5u6eB01 23 May, 2017 2.170.40.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
A0A0M3KKW9 A0A0M3KKW9_9HIV1 Human immunodeficiency virus 1 clade A/E 93TH057 HIV-1 gp120 core
A0A0M3KKW9 A0A0M3KKW9_9HIV1 Human immunodeficiency virus 1 clade A/E 93TH057 HIV-1 gp120 core