PDB Information

PDB5U4X
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
TP-064, a potent and selective small molecule inhibitor of PRMT4 for multiple myeloma.
Nakayama, K., Szewczyk, M.M., Dela Sena, C., Wu, H., Dong, A., Zeng, H., Li, F., de Freitas, R.F., Eram, M.S., Schapira, M., Baba, Y., Kunitomo, M., Cary, D.R., Tawada, M., Ohashi, A., Imaeda, Y., Saikatendu, K.S., Grimshaw, C.E., Vedadi, M., Arrowsmith, C.H., Barsyte-Lovejoy, D., Kiba, A., Tomita, D., Brown, P.J.
Oncotarget
HeaderTransferase
Released2016-12-06
Resolution1.880
CATH Insert Date25 Dec, 2016

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 26 Dec, 2016 Chopped
B 26 Dec, 2016 Chopped
C 26 Dec, 2016 Chopped
D 26 Dec, 2016 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5u4xA01 31 Dec, 2016 3.40.50.150 Assigned
5u4xA02 31 Dec, 2016 2.70.160.11 Assigned
5u4xB01 31 Dec, 2016 3.40.50.150 Assigned
5u4xB02 31 Dec, 2016 2.70.160.11 Assigned
5u4xC01 31 Dec, 2016 3.40.50.150 Assigned
5u4xC02 31 Dec, 2016 2.70.160.11 Assigned
5u4xD01 31 Dec, 2016 3.40.50.150 Assigned
5u4xD02 31 Dec, 2016 2.70.160.11 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q86X55 CARM1_HUMAN Homo sapiens Histone-arginine methyltransferase CARM1
Q86X55 CARM1_HUMAN Homo sapiens Histone-arginine methyltransferase CARM1
Q86X55 CARM1_HUMAN Homo sapiens Histone-arginine methyltransferase CARM1
Q86X55 CARM1_HUMAN Homo sapiens Histone-arginine methyltransferase CARM1