PDB Information

PDB5U2N
MethodX-RAY DIFFRACTION
Host OrganismMammalia
Gene SourceHomo sapiens
Primary Citation
Discovery and Characterization of Novel Nonsubstrate and Substrate NAMPT Inhibitors.
Wilsbacher, J.L., Cheng, M., Cheng, D., Trammell, S.A.J., Shi, Y., Guo, J., Koeniger, S.L., Kovar, P.J., He, Y., Selvaraju, S., Heyman, H.R., Sorensen, B.K., Clark, R.F., Hansen, T.M., Longenecker, K.L., Raich, D., Korepanova, A.V., Cepa, S., Towne, D.L., Abraham, V.C., Tang, H., Richardson, P.L., McLoughlin, S.M., Badagnani, I., Curtin, M.L., Michaelides, M.R., Maag, D., Buchanan, F.G., Chiang, G.G., Gao, W., Rosenberg, S.H., Brenner, C., Tse, C.
Mol. Cancer Ther.
HeaderTransferase/Transferase Inhibitor
Released2016-11-30
Resolution1.730
CATH Insert Date14 Nov, 2017

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5u2nA01 10 Dec, 2017 Holding pen
5u2nA02 10 Dec, 2017 3.20.20.70 Assigned
5u2nB01 10 Dec, 2017 Holding pen
5u2nB02 10 Dec, 2017 3.20.20.70 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P43490 NAMPT_HUMAN Homo sapiens Nicotinamide phosphoribosyltransferase
P43490 NAMPT_HUMAN Homo sapiens Nicotinamide phosphoribosyltransferase