PDB Information

PDB5U06
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery, Development, and Cellular Delivery of Potent and Selective Bicyclic Peptide Inhibitors of Grb7 Cancer Target.
Watson, G.M., Kulkarni, K., Sang, J., Ma, X., Gunzburg, M.J., Perlmutter, P., Wilce, M.C.J., Wilce, J.A.
J. Med. Chem.
HeaderSignaling Protein/Inhibitor
Released2016-11-22
Resolution2.100
CATH Insert Date17 Dec, 2017

PDB Images (13)

PDB Prints

PDB Chains (8)

Chain ID Date inserted into CATH CATH Status
A 17 Dec, 2017 Chopped
B 17 Dec, 2017 Chopped
C 17 Dec, 2017 Chopped
D 17 Dec, 2017 Chopped
L 17 Dec, 2017 Rejected
M 17 Dec, 2017 Rejected
N 17 Dec, 2017 Rejected
P 17 Dec, 2017 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5u06A00 22 Dec, 2017 3.30.505.10 Assigned
5u06B00 22 Dec, 2017 3.30.505.10 Assigned
5u06C00 22 Dec, 2017 3.30.505.10 Assigned
5u06D00 22 Dec, 2017 3.30.505.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q14451 GRB7_HUMAN Homo sapiens Growth factor receptor-bound protein 7
Q14451 GRB7_HUMAN Homo sapiens Growth factor receptor-bound protein 7
Q14451 GRB7_HUMAN Homo sapiens Growth factor receptor-bound protein 7
Q14451 GRB7_HUMAN Homo sapiens Growth factor receptor-bound protein 7