PDB Information

PDB5TMK
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHomo sapiens
Primary Citation
Optimization of 3,5-Disubstitued Piperidine: Discovery of Non-Peptide mimetics as an Orally Active Renin Inhibitor
Tokuhara, H., Imaeda, Y., Fukase, Y., Iwanaga, K., Taya, N., Watanabe, K., Kanagawa, R., Matsuda, K., Kajimoto, Y., Kusumoto, K., Kondo, M., Snell, G.P., Behnke, C.A., Kuroita, T.
To be published
HeaderHydrolase/Hydrolase Inhibitor
Released2016-10-13
Resolution2.650
CATH Insert Date14 Nov, 2017

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5tmkA01 10 Dec, 2017 2.40.70.10 Assigned
5tmkA02 10 Dec, 2017 2.40.70.10 Assigned
5tmkB01 10 Dec, 2017 2.40.70.10 Assigned
5tmkB02 10 Dec, 2017 2.40.70.10 Assigned

UniProtKB Entries (0)

Accession Gene ID Taxon Description