PDB 5teg
PDB Information
| PDB | 5TEG |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Turning a Substrate Peptide into a Potent Inhibitor for the Histone Methyltransferase SETD8.
ACS Med Chem Lett
|
| Header | Transferase |
| Released | 2016-09-21 |
| Resolution | 1.300 |
| CATH Insert Date | 08 Jan, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 09 Jan, 2017 | Chopped |
| B | 09 Jan, 2017 | Chopped |
| D | 09 Jan, 2017 | Rejected |
| E | 09 Jan, 2017 | Rejected |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5tegA00 | 16 Feb, 2017 | 2.170.270.10 | Assigned |
| 5tegB00 | 16 Feb, 2017 | 2.170.270.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P62805 | H4_HUMAN | Homo sapiens | Histone H4 |
| Q9NQR1 | KMT5A_HUMAN | Homo sapiens | N-lysine methyltransferase KMT5A |
| Q9NQR1 | KMT5A_HUMAN | Homo sapiens | N-lysine methyltransferase KMT5A |
| P62805 | H4_HUMAN | Homo sapiens | Histone H4 |
