PDB Information

PDB5TA4
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Potent Cyclophilin Inhibitors Based on the Structural Simplification of Sanglifehrin A.
Steadman, V.A., Pettit, S.B., Poullennec, K.G., Lazarides, L., Keats, A.J., Dean, D.K., Stanway, S.J., Austin, C.A., Sanvoisin, J.A., Watt, G.M., Fliri, H.G., Liclican, A.C., Jin, D., Wong, M.H., Leavitt, S.A., Lee, Y.J., Tian, Y., Frey, C.R., Appleby, T.C., Schmitz, U., Jansa, P., Mackman, R.L., Schultz, B.E.
J. Med. Chem.
HeaderIsomerase/Isomerase Inhibitor
Released2016-09-09
Resolution1.500
CATH Insert Date07 May, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5ta4A00 21 May, 2017 2.40.100.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P62937 PPIA_HUMAN Homo sapiens Peptidyl-prolyl cis-trans isomerase A