PDB 5t23
PDB Information
| PDB | 5T23 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Insect cell expression vector pTIE1 |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett.
|
| Header | Transferase |
| Released | 2016-08-23 |
| Resolution | 2.780 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (7)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Chopped |
CATH Domains (5)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5t23A01 | 20 May, 2017 | 3.10.20.90 | Assigned |
| 5t23A02 | 20 May, 2017 | 2.60.40.150 | Assigned |
| 5t23A03 | 20 May, 2017 | 1.25.40.70 | Assigned |
| 5t23A04 | 20 May, 2017 | 3.30.1010.10 | Assigned |
| 5t23A05 | 20 May, 2017 | 1.10.1070.11 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P48736 | PK3CG_HUMAN | Homo sapiens | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
