PDB 5swr
PDB Information
| PDB | 5SWR |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Identification of allosteric binding sites for PI3K alpha oncogenic mutant specific inhibitor design.
Bioorg. Med. Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2016-08-08 |
| Resolution | 3.310 |
| CATH Insert Date | 07 May, 2017 |
PDB Images (5)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 May, 2017 | Holding pen |
| B | 08 May, 2017 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5swrB01 | 14 Nov, 2017 | Holding pen | |
| 5swrB02 | 14 Nov, 2017 | 1.10.287.1490 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P27986 | P85A_HUMAN | Homo sapiens | Phosphatidylinositol 3-kinase regulatory subunit alpha |
| P42336 | PK3CA_HUMAN | Homo sapiens | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
