PDB 5qii
PDB Information
PDB | 5QII |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli BL21(DE3) |
Gene Source | Homo sapiens |
Primary Citation | Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11 beta-Hydroxysteroid Dehydrogenase Type 1 (11 beta-HSD-1).
ACS Med Chem Lett
|
Header | Oxidoreductase/Oxidoreductase Inhibitor |
Released | 2018-07-03 |
Resolution | 2.450 |
CATH Insert Date | 23 Dec, 2018 |
PDB Images (9)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 23 Dec, 2018 | Chopped |
B | 23 Dec, 2018 | Chopped |
D | 23 Dec, 2018 | Chopped |
E | 23 Dec, 2018 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5qiiA00 | 26 Dec, 2018 | 3.40.50.720 | Assigned |
5qiiB00 | 26 Dec, 2018 | 3.40.50.720 | Assigned |
5qiiD01 | 26 Dec, 2018 | 3.40.50.720 | Assigned |
5qiiE00 | 26 Dec, 2018 | 3.40.50.720 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |
P28845 | DHI1_HUMAN | Homo sapiens | Corticosteroid 11-beta-dehydrogenase isozyme 1 |