PDB Information

PDB5OT5
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Second-generation CK2 alpha inhibitors targeting the alpha D pocket.
Iegre, J., Brear, P., De Fusco, C., Yoshida, M., Mitchell, S.L., Rossmann, M., Carro, L., Sore, H.F., Hyvonen, M., Spring, D.R.
Chem Sci
HeaderTransferase
Released2017-08-21
Resolution1.630
CATH Insert Date03 Jun, 2018

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5ot5A01 27 Jun, 2018 1.10.510.10 Assigned
5ot5A02 27 Jun, 2018 3.30.200.20 Assigned
5ot5B01 27 Jun, 2018 1.10.510.10 Assigned
5ot5B02 27 Jun, 2018 3.30.200.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha