PDB 5o3i
PDB Information
| PDB | 5O3I |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli BL21 |
| Gene Source | Homo sapiens |
| Primary Citation | Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition.
Chem Sci
|
| Header | Transcription |
| Released | 2017-05-23 |
| Resolution | 1.200 |
| CATH Insert Date | 03 Jun, 2018 |
PDB Images (3)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 03 Jun, 2018 | Chopped |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5o3iA00 | 27 Jun, 2018 | 1.20.920.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P25440 | BRD2_HUMAN | Homo sapiens | Bromodomain-containing protein 2 |
