PDB Information

PDB5N20
MethodX-RAY DIFFRACTION
Host OrganismKomagataella pastoris
Gene SourceHomo sapiens
Primary Citation
Discovery of Pyrazolo[1,5-a]pyrimidine B-Cell Lymphoma 6 (BCL6) Binders and Optimization to High Affinity Macrocyclic Inhibitors.
McCoull, W., Abrams, R.D., Anderson, E., Blades, K., Barton, P., Box, M., Burgess, J., Byth, K., Cao, Q., Chuaqui, C., Carbajo, R.J., Cheung, T., Code, E., Ferguson, A.D., Fillery, S., Fuller, N.O., Gangl, E., Gao, N., Grist, M., Hargreaves, D., Howard, M.R., Hu, J., Kemmitt, P.D., Nelson, J.E., O'Connell, N., Prince, D.B., Raubo, P., Rawlins, P.B., Robb, G.R., Shi, J., Waring, M.J., Whittaker, D., Wylot, M., Zhu, X.
J. Med. Chem.
HeaderTransferase
Released2017-02-06
Resolution1.380
CATH Insert Date21 May, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 22 May, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5n20A00 06 Nov, 2017 3.30.710.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P41182 BCL6_HUMAN Homo sapiens B-cell lymphoma 6 protein