PDB Information

PDB5MWH
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-based discovery of selective BRPF1 bromodomain inhibitors.
Zhu, J., Zhou, C., Caflisch, A.
Eur J Med Chem
HeaderDna Binding Protein
Released2017-01-18
Resolution1.650
CATH Insert Date03 Jun, 2018

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Jun, 2018 Chopped
B 03 Jun, 2018 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5mwhA00 27 Jun, 2018 1.20.920.10 Assigned
5mwhB00 27 Jun, 2018 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P55201 BRPF1_HUMAN Homo sapiens Peregrin
P55201 BRPF1_HUMAN Homo sapiens Peregrin