PDB Information

PDB5LWP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of phenoxyindazoles and phenylthioindazoles as ROR gamma inverse agonists.
Ouvry, G., Bouix-Peter, C., Ciesielski, F., Chantalat, L., Christin, O., Comino, C., Duvert, D., Feret, C., Harris, C.S., Lamy, L., Luzy, A.P., Musicki, B., Orfila, D., Pascau, J., Parnet, V., Perrin, A., Pierre, R., Polge, G., Raffin, C., Rival, Y., Taquet, N., Thoreau, E., Hennequin, L.F.
Bioorg.Med.Chem.Lett.
HeaderTranscription
Released2016-09-19
Resolution2.400
CATH Insert Date27 Nov, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Nov, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5lwpA00 01 Dec, 2016 1.10.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma