PDB Information

PDB5LSX
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Structure of the Epigenetic Oncogene MMSET and Inhibition by N-Alkyl Sinefungin Derivatives.
Tisi, D., Chiarparin, E., Tamanini, E., Pathuri, P., Coyle, J.E., Hold, A., Holding, F.P., Amin, N., Martin, A.C., Rich, S.J., Berdini, V., Yon, J., Acklam, P., Burke, R., Drouin, L., Harmer, J.E., Jeganathan, F., van Montfort, R.L., Newbatt, Y., Tortorici, M., Westlake, M., Wood, A., Hoelder, S., Heightman, T.D.
ACS Chem. Biol.
HeaderTransferase
Released2016-09-05
Resolution2.900
CATH Insert Date16 Oct, 2016

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 17 Oct, 2016 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5lsxA00 22 Oct, 2016 2.170.270.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9BYW2 SETD2_HUMAN Homo sapiens Histone-lysine N-methyltransferase SETD2