PDB Information

PDB5LBQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21
Gene SourceHomo sapiens
Primary Citation
Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural features.
Speranzini, V., Rotili, D., Ciossani, G., Pilotto, S., Marrocco, B., Forgione, M., Lucidi, A., Forneris, F., Mehdipour, P., Velankar, S., Mai, A., Mattevi, A.
Sci Adv
HeaderOxidoreductase/Repressor
Released2016-06-16
Resolution3.300
CATH Insert Date09 Oct, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Oct, 2016 Chopped
B 10 Oct, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5lbqA01 15 Oct, 2016 1.10.10.10 Assigned
5lbqA02 15 Oct, 2016 Holding pen
5lbqA03 15 Oct, 2016 1.10.287.80 Assigned
5lbqB00 15 Oct, 2016 1.20.58.1880 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9UKL0 RCOR1_HUMAN Homo sapiens REST corepressor 1
O60341 KDM1A_HUMAN Homo sapiens Lysine-specific histone demethylase 1A