PDB Information

PDB5KZ8
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure guided design of a series of selective pyrrolopyrimidinone MARK inhibitors.
Katz, J.D., Haidle, A., Childers, K.K., Zabierek, A.A., Jewell, J.P., Hou, Y., Altman, M.D., Szewczak, A., Chen, D., Harsch, A., Hayashi, M., Warren, L., Hutton, M., Nuthall, H., Su, H.P., Munshi, S., Stanton, M.G., Davies, I.W., Munoz, B., Northrup, A.
Bioorg. Med. Chem. Lett.
HeaderTransferase/Transferase Inhibitor
Released2016-07-23
Resolution3.210
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Holding pen
B 14 Nov, 2017 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q7KZI7 MARK2_HUMAN Homo sapiens Serine/threonine-protein kinase MARK2
Q7KZI7 MARK2_HUMAN Homo sapiens Serine/threonine-protein kinase MARK2