PDB Information

PDB5KOT
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHomo sapiens
Primary Citation
Discovery of TAK-272: A Novel, Potent and Orally Active Renin Inhibitor
Imaeda, Y., Tokuhara, H., Fukase, Y., Kanagawa, R., Kajimoto, Y., Kusumoto, K., Kondo, M., Snell, G.P., Behnke, C.A., Kuroita, T.
To be published
HeaderHydrolase/Hydrolase Inhibitor
Released2016-07-01
Resolution2.100
CATH Insert Date14 Nov, 2017

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5kotA01 10 Dec, 2017 2.40.70.10 Assigned
5kotA02 10 Dec, 2017 2.40.70.10 Assigned
5kotB01 10 Dec, 2017 2.40.70.10 Assigned
5kotB02 10 Dec, 2017 2.40.70.10 Assigned

UniProtKB Entries (0)

Accession Gene ID Taxon Description