PDB 5kos
PDB Information
PDB | 5KOS |
Method | X-RAY DIFFRACTION |
Host Organism | Homo sapiens |
Gene Source | Homo sapiens |
Primary Citation | Discovery of TAK-272: A Novel, Potent, and Orally Active Renin Inhibitor.
Acs Med.Chem.Lett.
|
Header | Hydrolase/Hydrolase Inhibitor |
Released | 2016-07-01 |
Resolution | 2.410 |
CATH Insert Date | 27 Nov, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 28 Nov, 2016 | Chopped |
B | 28 Nov, 2016 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5kosA01 | 01 Dec, 2016 | 2.40.70.10 | Assigned |
5kosA02 | 01 Dec, 2016 | 2.40.70.10 | Assigned |
5kosB01 | 01 Dec, 2016 | 2.40.70.10 | Assigned |
5kosB02 | 01 Dec, 2016 | 2.40.70.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P00797 | RENI_HUMAN | Homo sapiens | Renin |
P00797 | RENI_HUMAN | Homo sapiens | Renin |