PDB 5kj0

PDB Information

PDB5KJ0
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHomo sapiens
Primary Citation
Assessment of Bromodomain Target Engagement by a Series of BI2536 Analogues with Miniaturized BET-BRET.
Koblan, L.W., Buckley, D.L., Ott, C.J., Fitzgerald, M.E., Ember, S.W., Zhu, J.Y., Liu, S., Roberts, J.M., Remillard, D., Vittori, S., Zhang, W., Schonbrunn, E., Bradner, J.E.
ChemMedChem
HeaderTranscription/Inhibitor
Released2016-06-17
Resolution1.510
CATH Insert Date14 Nov, 2017

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5kj0A01 10 Dec, 2017 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4