PDB 5kit
PDB Information
| PDB | 5KIT |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Minimizing CYP2C9 Inhibition of Exposed-Pyridine NAMPT (Nicotinamide Phosphoribosyltransferase) Inhibitors.
J.Med.Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2016-06-17 |
| Resolution | 1.600 |
| CATH Insert Date | 16 Oct, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 17 Oct, 2016 | Chopped |
| B | 17 Oct, 2016 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 5kitA01 | 21 Oct, 2016 | Holding pen | |
| 5kitA02 | 21 Oct, 2016 | 3.20.20.70 | Assigned |
| 5kitB01 | 22 Oct, 2016 | Holding pen | |
| 5kitB02 | 22 Oct, 2016 | 3.20.20.70 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P43490 | NAMPT_HUMAN | Homo sapiens | Nicotinamide phosphoribosyltransferase |
| P43490 | NAMPT_HUMAN | Homo sapiens | Nicotinamide phosphoribosyltransferase |
