PDB Information

PDB5KGT
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium bovis (strain ATCC BAA-935 / AF2122/97)
Primary Citation
Structure-Based Optimization of Pyridoxal 5'-Phosphate-Dependent Transaminase Enzyme (BioA) Inhibitors that Target Biotin Biosynthesis in Mycobacterium tuberculosis.
Liu, F., Dawadi, S., Maize, K.M., Dai, R., Park, S.W., Schnappinger, D., Finzel, B.C., Aldrich, C.C.
J. Med. Chem.
HeaderTransferase/Transferase Inhibitor
Released2016-06-13
Resolution2.250
CATH Insert Date14 Nov, 2017

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped
B 14 Nov, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5kgtA01 10 Dec, 2017 3.90.1150.10 Assigned
5kgtA02 10 Dec, 2017 3.40.640.10 Assigned
5kgtB01 10 Dec, 2017 3.90.1150.10 Assigned
5kgtB02 10 Dec, 2017 3.40.640.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P0A4X7 BIOA_MYCBO Mycobacterium tuberculosis variant bovis AF2122/97 Adenosylmethionine-8-amino-7-oxononanoate aminotransferase
P0A4X7 BIOA_MYCBO Mycobacterium tuberculosis variant bovis AF2122/97 Adenosylmethionine-8-amino-7-oxononanoate aminotransferase