PDB Information

PDB5J6S
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Crystal Structures of ERAP2 Complexed with Inhibitors Reveal Pharmacophore Requirements for Optimizing Inhibitor Potency.
Mpakali, A., Giastas, P., Deprez-Poulain, R., Papakyriakou, A., Koumantou, D., Gealageas, R., Tsoukalidou, S., Vourloumis, D., Mavridis, I.M., Stratikos, E., Saridakis, E.
ACS Med Chem Lett
HeaderHydrolase
Released2016-04-05
Resolution2.800
CATH Insert Date07 May, 2017

PDB Images (11)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5j6sA01 12 May, 2017 2.60.40.1730 Assigned
5j6sA02 12 May, 2017 1.10.390.10 Assigned
5j6sA03 12 May, 2017 2.60.40.1910 Assigned
5j6sA04 12 May, 2017 1.25.50.20 Assigned
5j6sB01 12 May, 2017 2.60.40.1730 Assigned
5j6sB02 12 May, 2017 1.10.390.10 Assigned
5j6sB03 12 May, 2017 2.60.40.1910 Assigned
5j6sB04 12 May, 2017 1.25.50.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q6P179 ERAP2_HUMAN Homo sapiens Endoplasmic reticulum aminopeptidase 2
Q6P179 ERAP2_HUMAN Homo sapiens Endoplasmic reticulum aminopeptidase 2