PDB Information

PDB5J1V
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structure.
Esvan, Y.J., Zeinyeh, W., Boibessot, T., Nauton, L., Thery, V., Knapp, S., Chaikuad, A., Loaec, N., Meijer, L., Anizon, F., Giraud, F., Moreau, P.
Eur.J.Med.Chem.
HeaderTransferase
Released2016-03-29
Resolution2.520
CATH Insert Date15 May, 2016

PDB Images (9)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 16 May, 2016 Chopped
B 16 May, 2016 Chopped
C 16 May, 2016 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5j1vA01 30 Nov, 2016 3.30.200.20 Assigned
5j1vA02 30 Nov, 2016 1.10.510.10 Assigned
5j1vB01 30 Nov, 2016 3.30.200.20 Assigned
5j1vB02 30 Nov, 2016 1.10.510.10 Assigned
5j1vC00 29 Nov, 2016 Holding pen

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P49759 CLK1_HUMAN Homo sapiens Dual specificity protein kinase CLK1
P49759 CLK1_HUMAN Homo sapiens Dual specificity protein kinase CLK1
P49759 CLK1_HUMAN Homo sapiens Dual specificity protein kinase CLK1