PDB Information

PDB5ITD
MethodX-RAY DIFFRACTION
Host Organismunidentified baculovirus
Gene SourceHomo sapiens
Primary Citation
Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors.
Hoegenauer, K., Soldermann, N., Stauffer, F., Furet, P., Graveleau, N., Smith, A.B., Hebach, C., Hollingworth, G.J., Lewis, I., Gutmann, S., Rummel, G., Knapp, M., Wolf, R.M., Blanz, J., Feifel, R., Burkhart, C., Zecri, F.
Acs Med.Chem.Lett.
HeaderTransferase/Protein Transport/Inhibitor
Released2016-03-16
Resolution3.020
CATH Insert Date09 Oct, 2016

PDB Images (10)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 10 Oct, 2016 Chopped
B 10 Oct, 2016 Chopped

CATH Domains (7)

Domain ID Date inserted into CATH Superfamily CATH Status
5itdA01 12 Jul, 2018 Check for files
5itdA02 12 Jul, 2018 Check for files
5itdA03 12 Jul, 2018 Check for files
5itdA04 12 Jul, 2018 Check for files
5itdA05 12 Jul, 2018 Check for files
5itdB01 14 Nov, 2017 Holding pen
5itdB02 14 Nov, 2017 1.10.287.1490 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P27986 P85A_HUMAN Homo sapiens Phosphatidylinositol 3-kinase regulatory subunit alpha
P42336 PK3CA_HUMAN Homo sapiens Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform